First Organocatalytic Asymmetric Biginelli Reaction
نویسندگان
چکیده
منابع مشابه
The direct organocatalytic asymmetric mannich reaction: unmodified aldehydes as nucleophiles.
The unprecedented application of unmodified aldehydes as nucleophilic donors in direct catalytic asymmetric Mannich-type reactions is disclosed in a full account. Our efforts in broadening the applicability of chiral pyrrolidine-based catalysts in direct asymmetric Mannich-type reactions led to the highly diastereo- and enantioselective and concise synthesis of functionalized alpha- and beta-am...
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ژورنال
عنوان ژورنال: Synfacts
سال: 2007
ISSN: 1861-1958,1861-194X
DOI: 10.1055/s-2006-955665